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Rupatadine Fumarate
CAS No. 182349-12-8
Rupatadine Fumarate ( —— )
Catalog No. M12814 CAS No. 182349-12-8
Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 50MG | 49 | Get Quote |
|
| 100MG | 73 | Get Quote |
|
| 500MG | 163 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameRupatadine Fumarate
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NoteResearch use only, not for human use.
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Brief DescriptionRupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
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DescriptionRupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
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Synonyms——
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH1 receptor; PAFR
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number182349-12-8
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Formula Weight532.03
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Molecular FormulaC26H26ClN3·C4H4O4
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Purity>98%(HPLC)
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SolubilityEthanol: 13 mg/mL (24.43 mM); DMSO: 9 mg/mL (16.91 mM)
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SMILESCC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Merlos M, et al. J Pharmacol Exp Ther, 1997, 280(1), 114-12
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